Patent · US Expired

Nonpeptidyl integrin inhibitors having specificity for the GPII.sub.b III.sub.a receptor

US5674863A · kind A · utility

10Cited by
11References
7Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMay 26, 1995
Grant dateOct 7, 1997
Priority date
Expiry dateMay 26, 2015

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D267/14
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

A benzodiazepinedione derivative which acts as a nonpeptidyl platelet aggregation inhibitor is provided. This inhibitor potently inhibits fibrinogen binding to the GPII.sub.b III.sub.a receptor and is provided in therapeutic compositions for the treatment of diseases for which blocking platelet aggregation is indicated. These nonpeptidyl inhibitors are provided in combination with thrombolytics and anticoagulants.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.