Collagenase-1 and stromelysin-1 inhibitors, pharmaceutical compositions comprising same and methods of their use
US5932579A · kind A · utility
56Cited by
11References
13Claims
0Family size
Assignee
Inventors
Key dates
| Filing date | Jun 18, 1996 |
| Grant date | Aug 3, 1999 |
| Priority date | — |
| Expiry date | Jun 18, 2016 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07D241/08
- WIPO fieldOrganic fine chemistry
- WIPO sectorChemistry
Abstract
Novel inhibitors of metalloproteases, in particular collagenase-1 and stromelysin-1, are disclosed. Such compounds are useful in pharmaceutical compositions and methods for treating or controlling disease states or conditions which involve tissue breakdown, such as rheumatoid arthritis. ##STR1##
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.