Patent · US Expired

Camptothecin compounds with combined topoisomerase I inhibition and DNA alkylation properties

US5932588A · kind A · utility

7Cited by
23References
4Claims
0Family size

Assignee

Inventors

Key dates

Filing dateOct 8, 1997
Grant dateAug 3, 1999
Priority date
Expiry dateOct 8, 2017

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D491/22
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Camptothecin compounds having a --CH.sub.2 --L group are effective anti-tumor compounds. These compounds inhibit the enzyme topoisomerase I and DNA of associated topoisomerase I-DNA complexes.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.