Patent · US Expired

Vinyl-pyrrolidinone cephalosporins

US5981519A · kind A · utility

5Cited by
1References
65Claims
0Family size

Assignee

Inventors

Key dates

Filing dateDec 8, 1997
Grant dateNov 9, 1999
Priority date
Expiry dateDec 8, 2017

Classification

  • Technology area (CPC Y)Emerging Cross-Sectional Technologies
  • CPC primaryY02P20/55
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present invention relates to compounds having the formula ##STR1## wherein X, R.sup.1, R.sup.2, R.sup.3, R.sup.4, R.sup.5, R.sup.6, and R.sup.7 are as defined herein as well as readily hydrolyzable esters thereof, pharmaceutically acceptable salts of said compounds and hydrates of the compounds of formula I and of their esters and salts. These compounds have valuable pharmacological activity for the treatment and prophylaxis of infectious diseases, especially those caused by methicillin resistant Staphylococcus aureus (MRSA) and Pseudomonas aeruginosa.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.