Patent · US Expired

Serine protease inhibitors-cycloheptane derivatives

US6015791A · kind A · utility

14Cited by
6References
32Claims
0Family size

Assignee

Inventors

Key dates

Filing dateDec 4, 1997
Grant dateJan 18, 2000
Priority date
Expiry dateDec 4, 2017

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61K38/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention relates to certain substituted oxadiazole, thiadiazole, and triazoles, in particular those including a cycloheptane structure, that are useful as serine protease inhibitors, including inhibitors for human neutrophil elastase. Compounds of the invention are useful in treating conditions such as adult respiratory distress syndrome, septic shock, and multiple organ failure.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.