Patent · US Expired

Matrix metalloprotease inhibitors

US6037472A · kind A · utility

12Cited by
16References
15Claims
0Family size

Assignee

Inventors

Key dates

Filing dateNov 22, 1994
Grant dateMar 14, 2000
Priority date
Expiry dateNov 22, 2014

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07C2603/18
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Compounds of formula (I) ##STR1## and their pharmaceutically acceptable salts inhibit matrix metalloproteases, such as stromelysin, gelatinase, matrilysin and collagenase, and are useful in the treatment of mammals having disease-states alleviated by the inhibition of such matrix metalloproteases.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.