Inventor · Haverstraw, NY, US

Arlindo L. Castelhano

49Patents
15h-index
72Co-inventors
84Inventor score

Filing activity: Jul 1, 1985 → Aug 26, 2022

Most-cited inventions

PatentTitleAreaCited byStatus
US5932595A Matrix metalloprotease inhibitors Chemistry; Metallurgy 62 Expired
US6680324B2 Compounds specific to adenosine A1 receptors and uses thereof Human Necessities 43 Expired
US6680322B2 Compounds specific to adenosine A1 receptors and uses thereof Human Necessities 40 Expired
US6008243A Metalloproteinase inhibitors, pharmaceutical compositions containing them, and their use Human Necessities 33 Expired
US5998412A Sulfamide-metalloprotease inhibitors Chemistry; Metallurgy 33 Expired
US7485658B2 N-substituted pyrazolyl-amidyl-benzimidazolyl c-Kit inhibitors Chemistry; Metallurgy 31 Expired
US4912120A 3,5-substituted 4,5-dihydroisoxazoles as transglutaminase inhibitors Chemistry; Metallurgy 27 Expired
US6143744A Sulfamide-metalloprotease inhibitors Chemistry; Metallurgy 27 Expired
US4929630A Transglutaminase inhibitors Chemistry; Metallurgy 26 Expired
US6916804B2 Pyrimidine A2b selective antagonist compounds, their synthesis and use Chemistry; Metallurgy 25 Expired
US7504407B2 Compounds specific to adenosine A1 and A3 receptors and uses thereof Human Necessities 22 Expired
US6800633B2 Pyrrolo[2,3d]pyrimidine compositions and their use Human Necessities 19 Expired
US6376506B1 Sulfamide-metalloprotease inhibitors Chemistry; Metallurgy 18 Expired
US6130220A Sulfamide-metalloprotease inhibitors Chemistry; Metallurgy 17 Expired
US6686366B1 Compounds specific to adenosine A3 receptor and uses thereof Human Necessities 15 Expired
US4970297A Transglutaminase inhibitors Emerging Cross-Sectional Technologies 15 Expired
US6673802B2 Compounds specific to adenosine A3 receptor and uses thereof Human Necessities 13 Expired
US6037472A Matrix metalloprotease inhibitors Chemistry; Metallurgy 12 Expired
US6878716B1 Compounds specific to adenosine A1 receptor and uses thereof Human Necessities 11 Expired
US6664252B2 4-aminopyrrolo[2,3-d]pyrimidine compounds specific to adenosine A2a receptor and uses thereof Human Necessities 11 Expired
US7501407B2 Pyrimidine A2B selective antagonist compounds, their synthesis and use Chemistry; Metallurgy 8 Expired
US7160890B2 Compounds specific to adenosine A3 receptor and uses thereof Chemistry; Metallurgy 7 Expired
US7429574B2 4-heterocyclo-pyrrolo[2,3d] pyrimidine compositions and their use Human Necessities 5 Expired
US7662844B2 Naphthylene derivatives as cytochrome P450 inhibitors Chemistry; Metallurgy 5 Expired
US6495699B2 Metalloproteinase inhibitors, pharmaceutical compositions containing them, and their use Human Necessities 5 Expired

Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.