Patent · US Expired

Methods of O-demethylation and N-deprotection

US6395900B1 · kind B1 · utility

16Cited by
0References
10Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJun 29, 2001
Grant dateMay 28, 2002
Priority date
Expiry dateJun 29, 2021

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D489/12
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present invention provides a method for N-deprotecting an opioid compound, a method for N-deprotecting and O-demethylating an opioid compound, a method for O-demethylating an opioid compound, and a method for O-demethylating a nonpeptidic delta agonist compound or an opioid compound having a tertiary amide with no significant reaction at amide groups.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.