Patent · US Expired

Inhibitors of interleukin-1&bgr; converting enzyme

US6420522B1 · kind B1 · utility

55Cited by
4References
10Claims
0Family size

Assignee

Inventors

Key dates

Filing dateOct 29, 1999
Grant dateJul 16, 2002
Priority date
Expiry dateOct 29, 2019

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61K38/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention relates to novel classes of compounds which are inhibitors of interleukin-1&bgr; converting enzyme. The ICE inhibitors of this invention are characterized by specific structural and physicochemical features. This invention also relates to pharmaceutical compositions comprising these compounds. The compounds and pharmaceutical compositions of this invention are particularly well suited for inhibiting ICE activity and consequently, may be advantageously used as agents against interleukin-1 mediated diseases, including inflammatory diseases, autoimmune diseases and neurodegenerative diseases. This invention also relates to methods for inhibiting ICE activity and methods for treating interleukin-1 mediated diseases using the compounds and compositions of this invention.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.