Patent · US Expired

Isoindolines, method of use, and pharmaceutical compositions

US6476052B1 · kind B1 · utility

149Cited by
28References
28Claims
0Family size

Assignee

Inventors

Key dates

Filing dateAug 7, 2000
Grant dateNov 5, 2002
Priority date
Expiry dateAug 22, 2020

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61K47/42
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Substituted 1-oxo-2-(2,6-dioxopiperidin-3-yl)isoindolines are useful in treating inflammation, inflammatory disease, autoimmune disease, and oncogenic or cancerous conditions in a mammal. Typical embodiments are 1-oxo-2-(2,6-dioxopiperidin-3yl)4-aminoisoindoline and 1-oxo-2-(2,6-dioxo-3-methylpiperidin-3-yl)aminoisoindoline.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.