Pyridobenzodiazepine and pyridobenzoxazepine carboxyamide vasopressin agonists
US6620807B1 · kind B1 · utility
20Cited by
10References
10Claims
0Family size
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Key dates
| Filing date | Feb 1, 2000 |
| Grant date | Sep 16, 2003 |
| Priority date | — |
| Expiry date | Feb 1, 2020 |
Classification
- Technology area (CPC A)Human Necessities
- CPC primaryA61P7/00
- WIPO fieldOrganic fine chemistry
- WIPO sectorChemistry
Abstract
The present invention provides benzoheterocyclic carboxyamides, particularly pyridobenzodiazepine and pyridobenzoxazepine carboxyamides, of the general formula: wherein: W is O or NH, optionally substituted, as well as methods and pharmaceutical compositions utilizing these compounds for providing a temporary delay of urination or for the treatment of disorder which may be remedied or alleviated by vasopressin agonist activity, including diabetes insipidus, nocturnal enuresis, nocturia, urinary incontinence, bleeding or coagulation disorders.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.