Inventor · Princeton Junction, NJ, US

Amedeo A. Failli

94Patents
25h-index
77Co-inventors
91Inventor score

Filing activity: Sep 11, 1974 → Aug 11, 2006

Most-cited inventions

PatentTitleAreaCited byStatus
US5120842A Silyl ethers of rapamycin Human Necessities 289 Expired
US5177203A Rapamycin 42-sulfonates and 42-(N-carboalkoxy) sulfamates useful as immunosuppressive agents Chemistry; Metallurgy 203 Expired
US5130307A Aminoesters of rapamycin Human Necessities 171 Expired
US5023264A Rapamycin oximes Chemistry; Metallurgy 146 Expired
US5162333A Aminodiesters of rapamycin Chemistry; Metallurgy 125 Expired
US5252579A Macrocyclic immunomodulators Human Necessities 125 Expired
US5389639A Amino alkanoic esters of rapamycin Human Necessities 117 Expired
US5563145A Rapamycin 42-oximes and hydroxylamines Chemistry; Metallurgy 113 Expired
US5489680A Carbamates of rapamycin Human Necessities 100 Expired
US5373014A Rapamycin oximes Chemistry; Metallurgy 98 Expired
US5480988A Carbamates of rapamycin Human Necessities 93 Expired
US5420289A Substituted indole-, indene-, pyranoindole- and tetrahydrocarbazole-alkanoic acid derivatives as inhibitors of PLA.sub.2 and lipoxygenase Chemistry; Metallurgy 76 Expired
US5346893A Rapamycin 42-sulfonates and 42-(N-carbalkoxy) sulfamates useful as immunosuppressive agents Chemistry; Metallurgy 60 Expired
US5120726A Rapamycin hydrazones Chemistry; Metallurgy 59 Expired
US5446048A Rapamycin oximes Chemistry; Metallurgy 55 Expired
US5164399A Rapamycin pyrazoles Chemistry; Metallurgy 49 Expired
US5776967A Pyranoindole inhibitors of COX--2 Chemistry; Metallurgy 49 Expired
US5504204A Carbamates of rapamycin Human Necessities 48 Expired
US6713607B2 Effector proteins of Rapamycin Human Necessities 48 Expired
US5830911A Pyranoindole and tetrahydrocarbazole inhibitors of COX-2 Chemistry; Metallurgy 41 Expired
US5559227A Carbamates of rapaycin Human Necessities 41 Expired
US5229516A Substituted indole-, indene-, pyranoindole- and tetrahydrocarbazole-alkanoic acid derivatives as inhibitors of PLA2 and lipoxygenase Chemistry; Metallurgy 36 Expired
US7022699B2 Cyclohexenyl phenyl diazepines vasopressin and oxytocin receptor modulators Human Necessities 28 Expired
US6511974B1 Tricyclic vasopressin agonists Chemistry; Metallurgy 26 Expired
US6194407A Tricyclic pyrido vasopressin agonists Human Necessities 25 Expired

Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.