Patent · US Expired

Macrocyclic compounds and preparation methods thereof

US6660832B1 · kind B1 · utility

9Cited by
6References
31Claims
0Family size

Assignee

Inventors

Key dates

Filing dateAug 20, 1999
Grant dateDec 9, 2003
Priority date
Expiry dateAug 20, 2019

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D257/10
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present invention is directed to macrocyclic compounds of the formula (I) wherein Q, X, R1 and R5 are as defined herein. Compounds of the invention are useful for therapeutic and prophylactic treatment of bacterial infection in mammals. Solid phase synthetic procedures are provided effecting synthesis of the macrocyclic rings attached to a solid support.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.