Amine compounds and combinatorial libraries comprising same
US6750344B1 · kind B1 · utility
Assignee
Inventors
Key dates
| Filing date | Sep 5, 1997 |
| Grant date | Jun 15, 2004 |
| Priority date | — |
| Expiry date | Sep 5, 2017 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC40B40/00
- WIPO fieldMeasurement
- WIPO sectorInstruments
Abstract
The present invention provides monocyclic, bicyclic and oligomeric amine compounds with at least two sites of diversity. These compounds are formed from monocyclic scaffolds which can be cyclized to form bicyclic amine scaffolds. These can then be reacted with building blocks to form the amine compounds of the invention. This invention further provides libraries or monocyclic, bicyclic and oligomeric amine compounds. Also provided are methods for preparing monocyclic, bicyclic and oligomeric amine compounds and libraries thereof. The present invention also provides pharmaceutical compositions of the monocyclic, bicyclic and oligomeric amine compounds.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.