Patent · US Expired

Isoindole-imide compounds, compositions, and uses thereof

US7091353B2 · kind B2 · utility

85Cited by
28References
15Claims
0Family size

Assignee

Inventors

Key dates

Filing dateDec 21, 2001
Grant dateAug 15, 2006
Priority date
Expiry dateDec 21, 2021

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D409/14
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The invention relates to isoindole-imide compounds and pharmaceutically acceptable salts, hydrates, solvates, clathrates, enantiomers, diastereomers, racemates, or mixtures of stereoisomers thereof, pharmaceutical compositions comprising these isoindole-imide compounds, and methods for reducing the level of cytokines and their precursors in mammals. In particular, the invention pertains to isoindole-imide compounds that are potent inhibitors of the production of TNF-α in mammals. The isoindole-imides described herein are useful for treating or preventing diseases or disorders in mammals, for example, cancers, such as solid tumors and blood-born tumors; heart disease, such as congestive heart failure; osteoporosis; and genetic, inflammatory; allergic; and autoimmune diseases.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.