Pyrazoloanthrone and derivatives thereof as JNK inhibitors and compositions and methods related thereto
US7119114B1 · kind B1 · utility
10Cited by
4References
19Claims
0Family size
Assignee
Inventors
Key dates
| Filing date | Aug 18, 2000 |
| Grant date | Oct 10, 2006 |
| Priority date | — |
| Expiry date | Aug 18, 2020 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07D409/12
- WIPO fieldPharmaceuticals
- WIPO sectorChemistry
Abstract
Compounds having activity as selective inhibitors of JNK are disclosed The compounds of this invention are pyrazoloanthrone and derivatives thereof having the following structure:wherein R1 and R2 are as defined herein. Such compounds have utility in the treatment of a wide range of conditions that are responsive to JNK inhibition. Thus, methods of treating such conditions are also disclosed, as are pharmaceutical compositions containing one or more compounds of the above compounds.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.