Patent · US Expired

Heteroaryl substituted spirocyclic sulfamides for inhibition of gamma secretase

US7282513B2 · kind B2 · utility

4Cited by
3References
10Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMar 2, 2006
Grant dateOct 16, 2007
Priority date
Expiry dateMar 2, 2026

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D491/04
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Compounds of formula I are disclosed:in which X is a 5-membered heteroaryl ring and R is as defined herein. The compounds are inhibitors of the processing of APP by gamma-secretase, and hence are useful in the treatment or prevention of Alzheimer's disease.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.