Small molecule entry inhibitors
US7429677B2 · kind B2 · utility
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1References
4Claims
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Assignee
Inventors
Key dates
| Filing date | Mar 11, 2003 |
| Grant date | Sep 30, 2008 |
| Priority date | — |
| Expiry date | Jun 20, 2023 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07D333/38
- WIPO fieldOrganic fine chemistry
- WIPO sectorChemistry
Abstract
The present invention concerns a compound having the formula (I)a N-oxide form, a stereochemical isomer, racemic mixture, salt, prodrug, ester or metabolite thereof. It further relates to processes for their preparation as well as pharmaceutical compositions, their use as medicines, and diagnostic kits comprising them. The present invention also concerns combinations of the present entry inhibitors with anti-retroviral agents. It further relates to their use in assays as reference compounds or as reagents. The compounds of the present invention are useful for preventing or treating infection by HIV and for treating AIDS.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.