Inventor · Frederick, MD, US

Michael Eissenstat

26Patents
4h-index
26Co-inventors
59Inventor score

Filing activity: Sep 28, 2001 → Jan 11, 2016

Most-cited inventions

PatentTitleAreaCited byStatus
US9403789B2 Benzofuran-containing amino acid inhibitors of cytochrome P450 Chemistry; Metallurgy 19 Active
US6649651B1 Hexahydrofuro[2,3-B]furan-3-yl-n{3[(1,3-benzodioxol-5-ylsulfonyl)(isobutyl)amino]-1-benzyl-2-hydroxypropyl}carbamate as retroviral protease inhibitor Human Necessities 9 Expired
US7109230B2 Resistance-repellent retroviral protease inhibitors Emerging Cross-Sectional Technologies 6 Expired
US7285566B2 Resistance-repellent retroviral protease inhibitors Physics 4 Expired
US6613764B1 Aspartic protease inhibitors Chemistry; Metallurgy 4 Expired
US7157495B2 Hexahydrofuro[2,3-B]furan-3-YL-N-{3-[(1,3-benzodioxol-5-ylsulfonyl)(isobutyl)amino]-1-benzyl-2-hydroxypropyl}carbamate as retroviral protease inhibitor Human Necessities 3 Expired
US8673970B2 HIV protease inhibitor and cytochrome p450 inhibitor combinations Human Necessities 3 Active
US7981929B2 Benzofuran derived HIV protease inhibitors Human Necessities 3 Active
US8906647B2 Diamide inhibitors of cytochrome P450 Emerging Cross-Sectional Technologies 2 Active
US7507763B2 Resistance-repellent retroviral protease inhibitors Human Necessities 2 Active
US8048871B2 Compositions and methods for inhibiting cytochrome P450 Chemistry; Metallurgy 2 Active
US7378441B2 Resistance-repellent retroviral protease inhibitors Human Necessities 2 Expired
US8765667B2 HCV protease inhibitors Chemistry; Metallurgy 2 Active
US7807845B2 Resistance-repellent retroviral protease inhibitors Chemistry; Metallurgy 1 Active
US8389571B2 Benzofuran derived HIV protease inhibitors Human Necessities 1 Active
US9540354B2 Diamide inhibitors of cytochrome P450 Emerging Cross-Sectional Technologies 1 Active
US8791157B2 5-substituted benzofurans as inhibitors of cytochrome P450 2D6 Chemistry; Metallurgy 1 Active
US8481520B2 Compositions and methods for inhibiting cytochrome P450 Chemistry; Metallurgy 0 Active
US8569364B2 5-substituted benzofurans as inhibitors of cytochrome P450 2D6 Chemistry; Metallurgy 0 Active
US7429677B2 Small molecule entry inhibitors Chemistry; Metallurgy 0 Expired
US8952056B2 Methods for inhibiting drug degradation Human Necessities 0 Active
US8703700B2 Bimacrocylic HCV NS3 protease inhibitors Chemistry; Metallurgy 0 Active
US9604952B2 Compositions and methods for inhibiting cytochrome P450 2D6 Chemistry; Metallurgy 0 Active
US9849107B2 Compositions and methods for inhibiting cytochrome P450 Chemistry; Metallurgy 0 Active
US7132420B2 Aspartic protease inhibitors Chemistry; Metallurgy 0 Expired

Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.