Patent · US Active

Variable domain library and uses

US7785903B2 · kind B2 · utility

24Cited by
43References
23Claims
0Family size

Assignee

Inventors

Key dates

Filing dateApr 8, 2005
Grant dateAug 31, 2010
Priority date
Expiry dateSep 14, 2026

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07K2318/20
  • WIPO fieldBiotechnology
  • WIPO sectorChemistry

Abstract

The invention provides polypeptides comprising a variant heavy chain variable framework domain (VFR). In some embodiments, the amino acids defining the VFR form a loop of an antigen binding pocket. In an embodiment, the polypeptide is a variable domain of a monobody and has a variant VFR. The polypeptide may optionally comprise one or more complementary determining regions (CDRs) of antibody variable domains. In an embodiment, the polypeptide is a variable domain of a monobody and has a variant VFR and one or more variant CDRs. Libraries of polypeptides that include a plurality of different antibody variable domains generated by creating diversity in a VFR, and optionally, one or more CDRs are provided and may be used as a source for identifying novel antigen binding polypeptides that can be used therapeutically or as reagents. The invention also provides fusion polypeptides, compositions, and methods for generating and using the polypeptides and libraries.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.