Patent · US Active

Thiazolopyrimidines and their use as inhibitors of phosphatidylinositol-3 kinase

US8168633B2 · kind B2 · utility

5Cited by
6References
12Claims
0Family size

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Key dates

Filing dateJan 7, 2011
Grant dateMay 1, 2012
Priority date
Expiry dateJan 7, 2031

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P43/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Thiazolopyrimidine compounds of formula I, where W represents a thiazole ring, selectively inhibit the p110 delta subtype of PI3 Kinase (PI3K), and are useful for treating diseases and disorders arising from abnormal cell growth, function or behavior associated with PI3 kinase such as cancer, immune disorders, cardiovascular disease, viral infection, inflammation, metabolism/endocrine function disorders and neurological disorders.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.