Patent · US Active

c-Met modulators and method of use

US8178532B2 · kind B2 · utility

40Cited by
56References
3Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMay 24, 2007
Grant dateMay 15, 2012
Priority date
Expiry dateNov 8, 2029

Classification

  • Technology area (CPC Y)Emerging Cross-Sectional Technologies
  • CPC primaryY02A50/30
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention provides compounds for modulating protein kinase enzymatic activity for modulating cellular activities such as proliferation, differentiation, programmed cell death, migration and chemoinvasion. More specifically, the invention provides quinazolines and quinolines which inhibit, regulate, and/or modulate kinase receptor, particularly c-Met, KDF, c-Kit, flt-3 and flt-4, signal transduction pathways related to the changes in cellular activities as mentioned above, compositions which contain these compounds, and methods of using them to treat kinase-dependent diseases and conditions. The present invention also provides methods for making compounds as mentioned above, and compositions which contain these compounds.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.