Patent assignee · US · COMPANY

Exelixis, Inc.

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173Patents
137Active
173Granted
55Portfolio score

Filing activity: May 26, 1998 → Nov 25, 2024 · 70 expiring within 5 years

Most-cited patents

PatentTitleAreaCited byStatus
US7265131B2 Isoquinolinone derivatives and their use as therapeutic agents Chemistry; Metallurgy 136 Expired
US7579473B2 c-Met modulators and methods of use Emerging Cross-Sectional Technologies 63 Active
US6703491B1 Drosophila sequences Human Necessities 61 Expired
US7704995B2 Protein kinase modulators and methods of use Chemistry; Metallurgy 60 Expired
US8497284B2 C-met modulators and method of use Emerging Cross-Sectional Technologies 50 Active
US8877776B2 (L)-malate salt of N-(4-{[6,7-bis(methyloxy) quinolin-4-yl]oxy}phenyl)-N'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide Chemistry; Metallurgy 47 Active
US7999006B2 Methods of using MEK inhibitors Human Necessities 45 Active
US8067436B2 c-Met modulators and methods of use Emerging Cross-Sectional Technologies 44 Active
US7989622B2 Phosphatidylinositol 3-kinase inhibitors and methods of their use Emerging Cross-Sectional Technologies 43 Active
US8178532B2 c-Met modulators and method of use Emerging Cross-Sectional Technologies 40 Active
US7977345B2 c-MET modulators and method of use Chemistry; Metallurgy 39 Active
US8476298B2 c-Met modulators and method of use Emerging Cross-Sectional Technologies 37 Active
US9724342B2 C-met modulator pharmaceutical compositions Human Necessities 35 Active
US8673912B2 Crystalline Forms on N-[3-fluoro-4-({6-(methyloxy)-7-[(3-morpholin-4-ylpropyl)oxy]-quinolin-4-yl}oxy)phenyl]-N′-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide Human Necessities 33 Active
US7485634B2 Azepinoindole and pyridoindole derivatives as pharmaceutical agents Chemistry; Metallurgy 29 Expired
US8222256B2 Methods of using IGFIR and ABL kinase modulators Human Necessities 28 Active
US7803839B2 Azetidines as MEK inhibitors for the treatment of proliferative diseases Chemistry; Metallurgy 28 Active
US10034873B2 C-met modulator pharmaceutical compositions Human Necessities 27 Active
US9717720B2 Processes for preparing quinoline compounds and pharmaceutical compositions containing such compounds Chemistry; Metallurgy 26 Active
US10039757B2 C-Met modulator pharmaceutical compositions Human Necessities 26 Active
US9809549B2 Malate salt of N-(4-{[6,7-bis(methyloxy)quinolin-4-yl]oxy}phenyl)-N′(4-fluorophenyl)cyclopropane-1,1-dicarboxamide, and crystalline forms therof for the treatment of cancer Chemistry; Metallurgy 24 Active
US6511824B1 Nucleic acids and polypeptides of invertebrate TWIK channels and methods of use Human Necessities 21 Expired
US9365516B2 Process for preparing quinoline derivatives Chemistry; Metallurgy 21 Active
US6852290B2 Multi-well apparatus Emerging Cross-Sectional Technologies 21 Expired
US8642584B2 Method of using PI3K and MEK modulators Chemistry; Metallurgy 20 Active

Source: USPTO / EPO open patent data. Counts and citation impact are objective bibliographic measures.