Patent · US Active

8-anilinoimidazopyridines and their use as anti-cancer and/or anti-inflammatory agents

US8293763B2 · kind B2 · utility

1Cited by
0References
17Claims
0Family size

Assignee

Inventors

Key dates

Filing dateDec 18, 2008
Grant dateOct 23, 2012
Priority date
Expiry dateSep 18, 2029

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D487/04
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The invention relates to imidazopyridines of formula I with anti-cancer and/or anti-inflammatory activity and more specifically to imidazopyridines which inhibit MEK kinase activity. The invention provides compositions and methods useful for inhibiting abnormal cell growth or treating a hyperproliferative disorder, or treating an inflammatory disease in a mammal. The invention also relates to methods of using the compounds for in vitro, in situ, and in vivo diagnosis or treatment of mammalian cells, or associated pathological conditions.(Formula I)

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.