Patent · US Active

Biaryl-spiroaminooxazoline analogues as alpha 2C adrenergic receptor modulators

US8324213B2 · kind B2 · utility

0Cited by
8References
11Claims
0Family size

Assignee

Inventors

Key dates

Filing dateOct 6, 2009
Grant dateDec 4, 2012
Priority date
Expiry dateOct 6, 2029

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D519/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

In its many embodiments, the present invention provides a novel class of biaryi spiroaminooxazoline analogues as modulators of α2C adrenergic receptor agonists, methods of preparing such compounds, pharmaceutical compositions containing one or more such compounds, methods of preparing pharmaceutical formulations comprising one or more such compounds, and methods of treatment, prevention, inhibition, or amelioration of one or more conditions associated with the α2C adrenergic receptors using such compounds or pharmaceutical compositions.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.