Patent · US Active

5H-cyclopenta[D]pyrimidines as AKT protein kinase inhibitors

US8329709B2 · kind B2 · utility

10Cited by
2References
33Claims
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Key dates

Filing dateJan 9, 2009
Grant dateDec 11, 2012
Priority date
Expiry dateJan 9, 2029

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D487/04
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Compounds of Formula I are useful for inhibiting AKT protein kinases. Methods using compounds of Formula I and stereoisomers and pharmaceutically acceptable salts thereof, for in vitro, in situ, and in vivo diagnosis, prevention or treatment of such disorders in mammalian cells, or associated pathological conditions are disclosed. Formula (I).

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.