Patent · US Active

Process for the preparation of morpholinyl anthracycline derivatives

US8470984B2 · kind B2 · utility

23Cited by

9References

7Claims

0Family size

Assignee

NERVIANO MEDICAL SCIENCES S.R.L. · IT

Inventors

Michele Caruso · Milano, IT
Vittoria Lupi · Milano, IT
Matteo Salsa · Novara, IT

Key dates

Filing date	Dec 1, 2011
Grant date	Jun 25, 2013
Priority date	—
Expiry date	Mar 11, 2032

Classification

Technology area (CPC C)Chemistry; Metallurgy
CPC primaryC07H19/24
WIPO fieldOrganic fine chemistry
WIPO sectorChemistry

Abstract

The present invention provides a process for the preparation of a morpholinyl anthracycline derivative in good yields and purity, including 3′-deamino-3″-4′-anhydro-[2″(S)-methoxy-3″(R)-hydroxy-4″-morpholinyl]doxorubicin (1).

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.