Inventor · Milano, IT

Michele Caruso

40Patents
10h-index
48Co-inventors
75Inventor score

Filing activity: Mar 24, 1986 → Nov 1, 2018

Most-cited inventions

PatentTitleAreaCited byStatus
US5387578A New linker for bioactive agents Chemistry; Metallurgy 35 Expired
US5547667A Linker for bioactive agents Chemistry; Metallurgy 31 Expired
US8389697B2 Anthracycline derivative conjugates, process for their preparation and their use as antitumor compounds Chemistry; Metallurgy 26 Active
US9604980B2 Substituted pyrimidinyl and pyridinyl-pyrrolopyridinones, process for their preparation and their use as kinase inhibitors Human Necessities 24 Active
US8470984B2 Process for the preparation of morpholinyl anthracycline derivatives Chemistry; Metallurgy 23 Active
US6586428B2 Combined preparations comprising morpholine anthracyclines and anticancer agent Human Necessities 23 Expired
US6403563B1 Antitumor composition containing a synergistic combination of an anthracycline derivative with a camptothecin derivate Human Necessities 21 Expired
US8900589B2 Anthracycline derivative conjugates, process for their preparation and their use as antitumor compounds Chemistry; Metallurgy 19 Active
US4985548A 4-demethoxy-4-amino-anthracyclines Human Necessities 15 Expired
US5731313A Use of anthracyclinone derivatives in amyloidosis Chemistry; Metallurgy 11 Expired
US4965351A 4-demethoxy-4-amino-anthracyclines Human Necessities 10 Expired
US9695240B2 Anthracycline derivative conjugates, process for their preparation and their use as antitumor compounds Chemistry; Metallurgy 8 Active
US5998615A Anthracyclinone derivatives Chemistry; Metallurgy 8 Expired
US6096888A Anthracyclinone derivatives and their use in amyloidosis Chemistry; Metallurgy 7 Expired
US4684629A 3'-deamino-3'-hydroxy-4'-deoxy-4'-amino doxorubicin and related daunorubicin Human Necessities 7 Expired
US5532218A 3'-aziridino-anthracycline derivatives Chemistry; Metallurgy 6 Expired
US5985887A Aza-anthracyclinone derivatives Chemistry; Metallurgy 6 Expired
US5744454A Anthracycline derivatives Chemistry; Metallurgy 5 Expired
US6194422A Anthracycline derivatives Human Necessities 4 Expired
US6103700A Fluoro labelled anthracyclinone and anthracycline derivatives Chemistry; Metallurgy 3 Expired
US5496808A Mono and bis alkylamino-anthracyclines Chemistry; Metallurgy 3 Expired
US9527863B2 Thieno-indole moieties and methods of treating using the same Chemistry; Metallurgy 3 Active
US8227472B2 Substituted pyrrolo-pyrazole derivatives as kinase inhibitors Human Necessities 2 Active
US8426417B2 Substituted pyrrolo-pyrimidine derivatives, process for their preparation and their use as kinase inhibitors Chemistry; Metallurgy 1 Active
US9561290B2 Functionalized thieno-indole derivatives for the treatment of cancer Chemistry; Metallurgy 1 Active

Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.