Patent · US Active

Pyrazolo[1,5-a]pyridines as MARK inhibitors

US8518911B2 · kind B2 · utility

1Cited by
1References
19Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJul 27, 2009
Grant dateAug 27, 2013
Priority date
Expiry dateMay 11, 2030

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D417/14
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The invention encompasses pyrazolo[1,5-a]pyridine derivatives which selectively inhibit microtubule affinity regulating kinase (MARK) and are therefore useful for the treatment or prevention of Alzheimer's disease. Pharmaceutical compositions and methods of use are also included.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.