Patent · US Active

Tetrahydroquinoline derivatives

US8546427B2 · kind B2 · utility

0Cited by
2References
24Claims
0Family size

Assignee

Inventors

Key dates

Filing dateOct 13, 2011
Grant dateOct 1, 2013
Priority date
Expiry dateOct 13, 2031

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D401/12
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention relates to compounds according to formula (I)and pharmaceutically acceptable salts or esters thereof, wherein R1 to R7 have the significance given herein. The compounds are activators of AMP-activated protein kinase (AMPK) and are useful in the treatment or prophylaxis of diseases that are related to AMPK regulation, such as obesity, dyslipidemia, hyperglycemia, type 1 or type 2 diabetes and cancers.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.