Patent · US Active

Biaryl-spiroaminooxzaoline analogues as alpha 2C adrenergic receptor modulators

US8569312B2 · kind B2 · utility

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1References
11Claims
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Inventors

Key dates

Filing dateApr 4, 2013
Grant dateOct 29, 2013
Priority date
Expiry dateApr 4, 2033

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D519/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

In its many embodiments, the present invention provides a novel class of biaryl spiroaminooxazoline analogues as modulators of α2C adrenergic receptor agonists, methods of preparing such compounds, pharmaceutical compositions containing one or more such compounds, methods of preparing pharmaceutical formulations comprising one or more such compounds, and methods of treatment, prevention, inhibition, or amelioration of one or more conditions associated with the α2C adrenergic receptors using such compounds or pharmaceutical compositions.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.