Patent · US Active

Neprilysin inhibitors

US8586536B2 · kind B2 · utility

68Cited by
21References
26Claims
0Family size

Assignee

Inventors

Key dates

Filing dateDec 14, 2011
Grant dateNov 19, 2013
Priority date
Expiry dateJan 19, 2032

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D498/04
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

In one aspect, the invention relates to compounds having the formula:where R1-R6, a, b, and X are as defined in the specification, or a pharmaceutically acceptable salt thereof. These compounds have neprilysin inhibition activity. In another aspect, the invention relates to pharmaceutical compositions comprising such compounds; methods of using such compounds; and processes and intermediates for preparing such compounds.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.