Patent assignee · US · COMPANY

Theravance, Inc.

387Patents
272Active
387Granted
53Portfolio score

Filing activity: Feb 19, 1999 → Jul 8, 2013 · 197 expiring within 5 years

Most-cited patents

PatentTitleAreaCited byStatus
US6693202B1 Muscarinic receptor antagonists Chemistry; Metallurgy 138 Expired
US7858583B2 Process for purifying glycopeptide phosphonate derivatives Chemistry; Metallurgy 90 Active
US7141671B2 Biphenyl derivatives Physics 85 Expired
US6635764B2 Therapeutic ureas Chemistry; Metallurgy 81 Expired
US8513244B2 Neprilysin inhibitors Chemistry; Metallurgy 76 Active
US8449890B2 Neprilysin inhibitors Chemistry; Metallurgy 68 Active
US8586536B2 Neprilysin inhibitors Chemistry; Metallurgy 68 Active
US8481044B2 Neprilysin inhibitors Chemistry; Metallurgy 66 Active
US8563512B2 Neprilysin inhibitors Emerging Cross-Sectional Technologies 63 Active
US8686184B2 Neprilysin inhibitors Chemistry; Metallurgy 62 Active
US6670376B1 Aryl aniline &bgr;2 adrenergic receptor agonists Chemistry; Metallurgy 62 Expired
US6541669B1 &bgr;2-adrenergic receptor agonists Physics 59 Expired
US8691868B2 Neprilysin inhibitors Human Necessities 57 Active
US6656694B2 Method for identifying a ligand for a biological substrate Emerging Cross-Sectional Technologies 51 Expired
US6576793B1 &bgr;2-adrenergic receptor agonists Chemistry; Metallurgy 49 Expired
US7288657B2 Biphenyl compounds useful as muscarinic receptor antagonists Chemistry; Metallurgy 49 Expired
US7265133B2 Biphenyl compounds useful as muscarinic receptor antagonists Chemistry; Metallurgy 45 Expired
US6653323B2 Aryl aniline &bgr;2 adrenergic receptor agonists Chemistry; Metallurgy 44 Expired
US6747043B2 Alkoxy aryl &bgr;2 adrenergic receptor agonists Chemistry; Metallurgy 41 Expired
US7345060B2 Compounds having β2 adrenergic receptor agonist and muscarinic receptor antagonist activity Chemistry; Metallurgy 40 Expired
US7879896B2 Dual-acting imidazole antihypertensive agents Chemistry; Metallurgy 40 Active
US7456199B2 Biphenyl compounds useful as muscarinic receptor antagonists Human Necessities 37 Expired
US7279458B2 Cross-linked glycopeptide-cephalosporin antibiotics Chemistry; Metallurgy 36 Expired
US8013005B2 Dual-acting antihypertensive agents Chemistry; Metallurgy 36 Active
US7700777B2 Crystalline forms of a biphenyl compound Chemistry; Metallurgy 36 Active

Source: USPTO / EPO open patent data. Counts and citation impact are objective bibliographic measures.