Patent · US Active

Cycloalkyl-fused tetrahydroquinolines as CRTH2 receptor modulators

US8592383B2 · kind B2 · utility

4Cited by
4References
48Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJun 14, 2012
Grant dateNov 26, 2013
Priority date
Expiry dateJun 14, 2032

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D417/12
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The invention provides certain cycloalkyl-fused tetrahydroquinolines of the Formula (I),and their pharmaceutically acceptable salts and esters, wherein R1, R2, R7, R8, R8a, E, Y, Z, n, u, and t are as defined herein. The invention also provides pharmaceutical compositions comprising such compounds, and methods of using the compounds for treating diseases or conditions associated with uncontrolled or inappropriate stimulation of CRTH2 function.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.