Processes for preparing substituted pyrimidines
US8779127B2 · kind B2 · utility
23Cited by
58References
28Claims
0Family size
Assignee
Inventors
Key dates
| Filing date | Aug 15, 2012 |
| Grant date | Jul 15, 2014 |
| Priority date | — |
| Expiry date | Aug 15, 2032 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07D453/02
- WIPO fieldPharmaceuticals
- WIPO sectorChemistry
Abstract
The present invention provides a facile process for the preparation of tri- and tetra—substituted pyrimidines. The process is useful for preparing inhibitors of protein kinases, especially Aurora kinase. These inhibitors are useful for treating or lessening the severity of Aurora—mediated diseases or conditions.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.