Patent · US Active

Pharmaceutical compounds

US8802670B2 · kind B2 · utility

2Cited by
11References
12Claims
0Family size

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Inventors

Key dates

Filing dateApr 24, 2007
Grant dateAug 12, 2014
Priority date
Expiry dateOct 23, 2028

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D495/04
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Compounds of Formulae Ia and Ib, and stereoisomers, geometric isomers, tautomers, solvates, metabolites and pharmaceutically acceptable salts thereof, are useful for inhibiting lipid kinases including PI3K, and for treating disorders such as cancer mediated by lipid kinases. Methods of using compounds of Formula Ia and Ib for in vitro, in situ, and in vivo diagnosis, prevention or treatment of such disorders in mammalian cells, or associated pathological conditions, are disclosed.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.