Patent · US Active

5H-cyclopenta[d]pyrimidines as AKT protein kinase inhibitors

US8895566B2 · kind B2 · utility

1Cited by
6References
34Claims
0Family size

Assignees

Inventors

Key dates

Filing dateNov 15, 2012
Grant dateNov 25, 2014
Priority date
Expiry dateFeb 7, 2033

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D487/04
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Compounds of Formula I are useful for inhibiting AKT protein kinases. Methods of using compounds of Formula I and stereoisomers and pharmaceutically acceptable salts thereof, for in vitro, in situ, and in vivo diagnosis, prevention or treatment of such disorders in mammalian cells, or associated pathological conditions are disclosed.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.