Patent · US Active

Phosphatidylinositol 3-kinase inhibitors

US9221795B2 · kind B2 · utility

8Cited by
35References
59Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJun 13, 2014
Grant dateDec 29, 2015
Priority date
Expiry dateJun 13, 2034

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P37/06
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present disclosure provides phosphatidylinositol 3-kinase (PI3K) inhibitors of formula (I),or pharmaceutically acceptable salts or isomers thereof, in which n, m, R1, R2, R4, and R3 are as defined herein. These compounds are useful for treatment of conditions mediated by one or more PI3K isoforms, such as PI3Kδ. The present disclosure further provides pharmaceutical compositions that include a compound of formula (I), or pharmaceutically acceptable salts or isomers thereof, and methods of using these compounds and compositions to treat conditions mediated by one or more PI3K isoforms, such as PI3Kδ.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.