Patent · US Active

Heteroaryl pyridone and aza-pyridone compounds

US9238655B2 · kind B2 · utility

7Cited by
9References
8Claims
0Family size

Assignee

Inventors

Key dates

Filing dateSep 8, 2014
Grant dateJan 19, 2016
Priority date
Expiry dateSep 8, 2034

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07F7/1804
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Heteroaryl pyridone and aza-pyridone compounds are provided, including stereoisomers, tautomers, and pharmaceutically acceptable salts thereof, useful for inhibiting Btk kinase, and for treating immune disorders such as inflammation mediated by Btk kinase. Methods of using heteroaryl pyridone and aza-pyridone compounds for in vitro, in situ, and in vivo diagnosis, and treatment of such disorders in mammalian cells, or associated pathological conditions, are disclosed.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.