Patent · US Active

Aminopyrimidines as Syk inhibitors

US9290490B2 · kind B2 · utility

9Cited by
25References
25Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMay 4, 2012
Grant dateMar 22, 2016
Priority date
Expiry dateJul 8, 2032

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D417/14
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention provides novel pyrimidine amines of formula I which are potent inhibitors of spleen tyrosine kinase, and are useful in the treatment and prevention of diseases mediated by said enzyme, such as asthma, COPD, rheumatoid arthritis and cancer.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.