Patent · US Active

Processes for preparing JAK inhibitors and related intermediate compounds

US9290506B2 · kind B2 · utility

56Cited by
23References
1Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJan 9, 2015
Grant dateMar 22, 2016
Priority date
Expiry dateJan 9, 2035

Classification

  • Technology area (CPC Y)Emerging Cross-Sectional Technologies
  • CPC primaryY02P20/55
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present invention is related to processes for preparing chiral substituted pyrazolyl pyrrolo[2,3-d]pyrimidines of Formula III, and related synthetic intermediate compounds. The chiral substituted pyrazolyl pyrrolo[2,3-d]pyrimidines are useful as inhibitors of the Janus Kinase family of protein tyrosine kinases (JAKs) for treatment of inflammatory diseases, myeloproliferative disorders, and other diseases.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.