Patent · US Active

Process for making hydroxylated cyclopentylpyrimidine compounds

US9309204B2 · kind B2 · utility

7Cited by
3References
16Claims
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Key dates

Filing dateMay 17, 2013
Grant dateApr 12, 2016
Priority date
Expiry dateMay 17, 2033

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D403/04
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The invention provides new processes for making and purifying hydroxylated cyclopenta[d]pyrimidine compounds, which are useful for the treatment of diseases such as cancer as AKT protein kinase inhibitors, including the compound (S)-2-(4-chlorophenyl)-1-(4-((5R,7R)-7-hydroxy-5-methyl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)piperazin-1-yl)-3-(isopropylamino)propan-1-one.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.