Estrogen receptor modulators and uses thereof

US9399646B2 · kind B2 · utility

Assignee

• Genentech, Inc. · US

Inventors

• Nicholas D. Smith · San Diego, US
• Mehmet Kahraman · Village of La Jolla, US
• Steven P. Govek · San Diego, US
• Johnny Y. Nagasawa · San Diego, US
• Andiliy G. Lai · San Diego, US
• Jackaline D. Julien · Del Mar, US
• Mark R. Herbert · San Diego, US
• Celine Bonnefous · San Diego, US
• Karensa L. Douglas · San Diego, US

Key dates

• Filing date: Sep 15, 2011
• Grant date: Jul 26, 2016
• Expiry date: Feb 23, 2033

Classification

• Technology area (CPC C): Chemistry; Metallurgy
• CPC primary: C07D495/04
• WIPO field: Pharmaceuticals
• WIPO sector: Chemistry

Abstract

Described herein are compounds that are estrogen receptor modulators. Also described are pharmaceutical compositions and medicaments that include the compounds described herein, as well methods of using such estrogen receptor modulators, alone and in combination with other compounds, for treating diseases or conditions that are mediated or dependent upon estrogen receptors.