Patent · US Active

Pyrimidinones as PI3K inhibitors

US9434746B2 · kind B2 · utility

28Cited by
36References
25Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJan 2, 2014
Grant dateSep 6, 2016
Priority date
Expiry dateJan 2, 2034

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D513/04
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention provides pyrimidinones that modulate the activity of phosphoinositide 3-kinases (PI3Ks) and are useful in the treatment of diseases related to the activity of PI3Ks including, for example, inflammatory disorders, immune-based disorders, cancer, and other diseases.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.