Patent · US Active

Substituted bicyclic dihydropyrimidinones and their use as inhibitors of neutrophil elastase activity

US9475779B2 · kind B2 · utility

0Cited by
4References
14Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJul 27, 2015
Grant dateOct 25, 2016
Priority date
Expiry dateJul 27, 2035

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D405/06
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Substituted bicyclic dihydropyrimidinones of formula 1which are inhibitors of neutrophil elastase and useful as medicaments for the treatment of, inter alia, COPD. An exemplary compound is:

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.