Ralf Anderskewitz
48Patents
10h-index
55Co-inventors
78Inventor score
Filing activity: Jun 5, 1995 → Jun 6, 2017
Most-cited inventions
| Patent | Title | Area | Cited by | Status |
|---|---|---|---|---|
| US8987249B2 | Substituted 2-Aza-bicyclo[2.2.1]heptane-3-carboxylic acid (benzyl-cyano-methyl)-amides inhibitors of Cathepsin C | Emerging Cross-Sectional Technologies | 42 | Active |
| US9073869B2 | Method of using substituted 2-Aza-bicyclo[2.2.2]octane-3-carboxylic acid (benzyl-cyano-methyl)-amides inhibitors of cathepsin C | Chemistry; Metallurgy | 18 | Active |
| US8877775B2 | Substituted 2-aza-bicyclo[2.2.2]octane-3-carboxylic acid (benzyl-cyano-methyl)-amides inhibitors of cathepsin C | Chemistry; Metallurgy | 17 | Active |
| US8889708B2 | Substituted bicyclic 1-carboxylic-acid (benzyl-cyano-methyl)-amides inhibitors of cathepsin C | Emerging Cross-Sectional Technologies | 17 | Active |
| US10238633B2 | Methods for treating pulmonary emphysema using substituted 2-Aza-bicyclo[2.2.1]heptane-3-carboxylic acid (benzyl-cyano-methyl)-amides inhibitors of Cathepsin C | Emerging Cross-Sectional Technologies | 16 | Active |
| US9713606B2 | Methods for treating pulmonary emphysema using substituted 2-Aza-bicyclo[2.2.1]heptane-3-carboxylic acid (benzyl-cyano-methyl)-amides inhibitors of cathepsin C | Emerging Cross-Sectional Technologies | 16 | Active |
| US8871783B2 | Substituted 2-aza-bicyclo[2.2.1]heptane-3-carboxylic acid (cyano-methyl)-amides inhibitors of cathepsin C | Chemistry; Metallurgy | 15 | Active |
| US9440960B2 | Substituted oxetanes and their use as inhibitors of cathepsin C | Chemistry; Metallurgy | 15 | Active |
| US5731332A | Substituted benzamidine compounds which have useful pharmaceutical activity | Human Necessities | 14 | Expired |
| US6197824A | Benzamidine derivatives and the use thereof as medicaments with LTB4-antagonistic effect | Chemistry; Metallurgy | 11 | Expired |
| US6037377A | Amidine derivatives, the preparation and use thereof as medicaments with LTB4 antagonistic effect | Chemistry; Metallurgy | 10 | Expired |
| US5686496A | Chemical compound, the preparation thereof and its use in pharmaceutical compositions | Human Necessities | 9 | Expired |
| US6127423A | Phenylamidine derivatives, a process for preparing the same and their use as medicaments | Chemistry; Metallurgy | 7 | Expired |
| US6265612A | Benzamidine derivatives and the use thereof as medicaments with LTB4-antagonistic effect | Chemistry; Metallurgy | 6 | Expired |
| US6512000B1 | Aminocarbonyl-substituted benzimidazoles having tryptase-inhibitory activity | Chemistry; Metallurgy | 5 | Expired |
| US8637519B2 | Heterocycle-substituted piperazino-dihydrothienopyrimidines | Human Necessities | 5 | Active |
| US8754073B2 | Substituted piperazino-dihydrothienopyrimidines | Chemistry; Metallurgy | 5 | Active |
| US9440930B2 | Substituted bicyclic dihydropyrimidinones and their use as inhibitors of neutrophil elastase activity | Chemistry; Metallurgy | 4 | Active |
| US6855713B2 | Benzimidazole derivatives, a process for their manufacture and use as a medicine | Chemistry; Metallurgy | 3 | Expired |
| US6288277A | Benzylamine and phenylethylamine derivatives, processes for preparing the same and their use as medicaments | Chemistry; Metallurgy | 3 | Expired |
| US8791272B2 | Pyrazole compounds as CRTH2 antagonists | Chemistry; Metallurgy | 3 | Active |
| US6489365B1 | Amidine derivatives, the preparation and use thereof as medicaments with Itb4 antagonistic effect | Chemistry; Metallurgy | 3 | Expired |
| US6365584B1 | Arylysulphonamide-substituted benzimidazoles having tryptase-inhibiting activity | Chemistry; Metallurgy | 3 | Expired |
| US7544806B2 | Piperidine-substituted indoles-or heteroderivatives thereof | Chemistry; Metallurgy | 3 | Expired |
| US6291531A | LTB4 antagonist, processes for the preparation thereof and its use as a pharmaceutical composition | Chemistry; Metallurgy | 2 | Expired |
Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.