Pyrrol-1-yl benzoic acid derivatives useful as myc inhibitors
US9567301B2 · kind B2 · utility
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10Claims
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Key dates
| Filing date | Nov 1, 2013 |
| Grant date | Feb 14, 2017 |
| Priority date | — |
| Expiry date | Nov 1, 2033 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07D417/06
- WIPO fieldOrganic fine chemistry
- WIPO sectorChemistry
Abstract
The present invention provides compounds of Formula (I-A), (I-B), and (I-C), pharmaceutically acceptable salts thereof, and pharmaceutical compositions thereof. Compounds of the present invention are useful for inhibiting Myc (e.g., c-Myc) activity. The present invention further provides methods of using the compounds described herein for treating Myc-mediated disorders (e.g., cancer and other proliferative diseases). The present invention also provides assays for identifying Myc inhibitors.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.