Patent · US Active

Tetrahydronaphthyridine and related bicyclic compounds for inhibition of RORγ activity and the treatment of disease

US9657033B2 · kind B2 · utility

19Cited by
26References
44Claims
0Family size

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Key dates

Filing dateMay 7, 2013
Grant dateMay 23, 2017
Priority date
Expiry dateMay 7, 2033

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D471/04
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The invention provides tetrahydronaphthyridine and related compounds, pharmaceutical compositions, methods of inhibiting RORγ activity, reducing the amount of IL-17 in a subject, and treating immune disorders and inflammatory disorders using such tetrahydronaphthyridine and related compounds.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.