Patent · US Active

Process for making reverse transcriptase inhibitors

US9663490B2 · kind B2 · utility

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25Claims
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Inventors

Key dates

Filing dateDec 4, 2013
Grant dateMay 30, 2017
Priority date
Expiry dateDec 4, 2033

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P31/18
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present invention is directed to a novel process for synthesizing 3-(substituted phenoxy)-1-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl])-pyridin-2(1H)-one derivatives. The compounds synthesized by the processes of the invention are HIV reverse transcriptase inhibitors useful for inhibiting reverse transcriptase, HIV replication and the treatment of human immunodeficiency virus infection in humans.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.