Patent · US Active

Heteroaryl pyridone and aza-pyrodine compounds

US9782405B2 · kind B2 · utility

6Cited by
10References
14Claims
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Key dates

Filing dateNov 17, 2015
Grant dateOct 10, 2017
Priority date
Expiry dateNov 17, 2035

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07F7/1804
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Heteroaryl pyridone and aza-pyridone compounds are provided, including stereoisomers, tautomers, and pharmaceutically acceptable salts thereof, useful for inhibiting Btk kinase, and for treating immune disorders such as inflammation mediated by Btk kinase. Methods of using heteroaryl pyridone and aza-pyridone compounds for in vitro, in situ, and in vivo diagnosis, and treatment of such disorders in mammalian cells, or associated pathological conditions, are disclosed.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.